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| TEGASEROD MALEATE | ||
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PRODUCT IDENTIFICATION |
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| CAS NO. | 189188-57-6 |
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| EINECS NO. | ||
| FORMULA | C16H23N5O·C4H4O4 | |
| MOL WT. | 417.47 | |
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H.S. CODE |
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TOXICITY |
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| SYNONYMS | ||
| 3-(5-Methoxy-1H-indol-3-ylmethylene)-N-pentylcarbazimidamide hydrogen maleate; | ||
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CLASSIFICATION |
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PHYSICAL AND CHEMICAL PROPERTIES |
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| PHYSICAL STATE | white to off-white crystalline powder | |
| MELTING POINT | 152 - 155 C | |
| BOILING POINT | ||
| SPECIFIC GRAVITY | ||
| SOLUBILITY IN WATER | Practically insoluble | |
| pH | ||
| VAPOR DENSITY |
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| AUTOIGNITION |
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| NFPA RATINGS |
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REFRACTIVE INDEX |
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| FLASH POINT |
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| STABILITY |
Stable under ordinary conditions |
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APPLICATIONS |
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| Tegaserod is a medicine to increase bowel movement and used to treat short term IBS (irritable bowel syndrome), abdominal pain and discomfort, bloating, and constipation for women. The hydrogen maleate salt of tegaserod is a white to off-white crystalline powder; practicaly insoluble in water, slightly soluble in ethanol; melting point 152 - 153 C; administered orally. Chemical designation is 3-(5-methoxy-1H-indol-3-ylmethylene)-N-pentylcarbazimidamide hydrogen maleate. | ||
| SALES SPECIFICATION | ||
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APPEARANCE |
white to off-white crystalline powder | |
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IDENTIFICATION |
Complies Test A,B |
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| ASSAY |
99.0% min |
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LOSS ON DRYING |
1.0% max |
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RELATED SUBSTANCE |
0.5% max |
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HEAVY METALS |
20ppm max |
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| SULFATED ASH |
0.1% max |
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| TRANSPORTATION | ||
| PACKING |
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| HAZARD CLASS | ||
| UN NO. | ||
| OTHER INFORMATION | ||
| Hazard Symbols: n/a, Risk Phrases: 42/43, Safety Phrases: 22-36/37-45 | ||
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